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(S)-Timolol maleate
CAS No. 26921-17-5
(S)-Timolol maleate ( Timolol maleate )
产品货号. M13824 CAS No. 26921-17-5
A potent non-selective β-adrenergic receptor antagonist with Ki of 1.97 and 2 nM for β1 and β2 receptor, respectively.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 100MG | 获取报价 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称(S)-Timolol maleate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A potent non-selective β-adrenergic receptor antagonist with Ki of 1.97 and 2 nM for β1 and β2 receptor, respectively.
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产品描述A potent non-selective β-adrenergic receptor antagonist with Ki of 1.97 and 2 nM for β1 and β2 receptor, respectively.Hypertension Approved
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同义词Timolol maleate
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通路Angiogenesis
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靶点Adrenergic Receptor
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受体β1-adrenergicreceptor;β2-adrenergicreceptor
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研究领域Cardiovascular Disease
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适应症Hypertension
化学信息
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CAS Number26921-17-5
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分子量432.49
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分子式C17H28N4O7S
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 4.4 mg/mL
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SMILESCC(C)(C)NC[C@@H](COC1=NSN=C1N2CCOCC2)O.C(=C\C(=O)O)\C(=O)O
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化学全称2-Propanol, 1-[(1,1-dimethylethyl)amino]-3-[[4-(4-morpholinyl)-1,2,5-thiadiazol-3-yl]oxy]-, (2S)-, (2Z)-2-butenedioate (1:1)
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Mandagere AK, et al. J Med Chem. 2002;45(2):304-11.
2. Aggarwal D, et al. Int J Pharm. 2005 Feb 16;290(1-2):155-9.
3. Borok J, et al. Br J Dermatol. 2017 Aug 3. doi: 10.1111/bjd.15865.
2. Aggarwal D, et al. Int J Pharm. 2005 Feb 16;290(1-2):155-9.
3. Borok J, et al. Br J Dermatol. 2017 Aug 3. doi: 10.1111/bjd.15865.
产品手册
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